Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Wed Apr 02 02:58:31 GMT 2025
by
admin
on
Wed Apr 02 02:58:31 GMT 2025
|
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
66UL4XJJ3X
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
P43119
Created by
admin on Wed Apr 02 02:58:31 GMT 2025 , Edited by admin on Wed Apr 02 02:58:31 GMT 2025
|
PRIMARY | |||
|
66UL4XJJ3X
Created by
admin on Wed Apr 02 02:58:31 GMT 2025 , Edited by admin on Wed Apr 02 02:58:31 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_5 | 1_165 |
| 1_92 | 1_170 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_7 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
AGONIST -> TARGET |
EC50
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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|
AGONIST -> TARGET |
ACT-333679 is 37-fold more potent than selexipag towards prostacyclin IP receptor.
IC50
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
Assumed similar activity as prostaglandin E1
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AGONIST -> TARGET |
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AGONIST -> TARGET |
BINDING
IC50
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AGONIST -> TARGET |
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Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_383] | MECYSTEINE | RQ6L463N3B |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|
||||
| Molecular Formula | CHEMICAL |
|