U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 15:01:09 UTC 2023
Edited
by admin
on Sat Dec 16 15:01:09 UTC 2023
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
66UL4XJJ3X
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
PROSTACYCLIN RECEPTOR
Common Name English
PRIPR
Common Name English
PROSTAGLANDIN I2 RECEPTOR
Common Name English
Prostanoid IP receptor
Common Name English
Code System Code Type Description
UNIPROT
P43119
Created by admin on Sat Dec 16 15:01:10 UTC 2023 , Edited by admin on Sat Dec 16 15:01:10 UTC 2023
PRIMARY
FDA UNII
66UL4XJJ3X
Created by admin on Sat Dec 16 15:01:10 UTC 2023 , Edited by admin on Sat Dec 16 15:01:10 UTC 2023
PRIMARY
From To
1_5 1_165
1_92 1_170
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_7
Related Record Type Details
AGONIST -> TARGET
EC50
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
ACT-333679 is 37-fold more potent than selexipag towards prostacyclin IP receptor.
IC50
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
BINDING
IC50
AGONIST -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL