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Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 15:03:55 UTC 2023
Edited
by admin
on Sat Dec 16 15:03:55 UTC 2023
Protein Type REGULATOR PROTEIN
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
63L54VY2VT
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
APOPTOSIS REGULATOR BCL-X
Common Name English
BCL-XL
Common Name English
BCL2-L-1
Common Name English
BCL-2-LIKE PROTEIN 1
Common Name English
BCLX
Common Name English
B-CELL LYMPHOMA-EXTRA LARGE
Common Name English
Code System Code Type Description
FDA UNII
63L54VY2VT
Created by admin on Sat Dec 16 15:03:56 UTC 2023 , Edited by admin on Sat Dec 16 15:03:56 UTC 2023
PRIMARY
UNIPROT
Q07817
Created by admin on Sat Dec 16 15:03:56 UTC 2023 , Edited by admin on Sat Dec 16 15:03:56 UTC 2023
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
DEGRADER, SELECTIVE->TARGET
a von Hippel-Landau (VHL)-recruiting PROTAC; maximum degradation (Dmax) of 90.8%, and the degradation was dependent on both VHL and proteasome. MOLT-4 T-cell acute lymphoblastic leukemia (T-ALL) cells
DC50
INHIBITOR -> TARGET
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL