U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 03:35:12 GMT 2025
Edited
by admin
on Wed Apr 02 03:35:12 GMT 2025
Protein Type RECEPTOR
Protein Sub Type TYROSINE KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
5XEU95RN57
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ANAPLASTIC LYMPHOMA KINASE S1206Y
Common Name English
CD-246 S1206Y
Preferred Name English
ALK TYROSINE KINASE RECEPTOR S1206Y
Systematic Name English
CD246 S1206Y
Code English
ALK S1206Y MUTANT
Common Name English
Code System Code Type Description
UNIPROT
Q9UM73
Created by admin on Wed Apr 02 03:35:12 GMT 2025 , Edited by admin on Wed Apr 02 03:35:12 GMT 2025
PRIMARY
FDA UNII
5XEU95RN57
Created by admin on Wed Apr 02 03:35:12 GMT 2025 , Edited by admin on Wed Apr 02 03:35:12 GMT 2025
PRIMARY
WIKIPEDIA
ANAPLASTIC LYMPHOMA KINASE
Created by admin on Wed Apr 02 03:35:12 GMT 2025 , Edited by admin on Wed Apr 02 03:35:12 GMT 2025
PRIMARY
EC (ENZYME CLASS)
EC 2.7.10.1
Created by admin on Wed Apr 02 03:35:12 GMT 2025 , Edited by admin on Wed Apr 02 03:35:12 GMT 2025
PRIMARY
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_151
N 1_226
N 1_267
N 1_306
N 1_393
N 1_406
N 1_427
N 1_545
N 1_553
N 1_609
N 1_691
N 1_790
N 1_845
N 1_846
N 1_868
N 1_968
Related Record Type Details
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_1060] [1_1074] [1_1078] [1_1113] [1_1260] [1_1489] [1_1586] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL