U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
This repository is under review for potential modification in compliance with Administration directives.

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 16:59:35 GMT 2025
Edited
by admin
on Tue Apr 01 16:59:35 GMT 2025
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
5NJ22TAB5Y
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
PIM1
Preferred Name English
SERINE/THREONINE-PROTEIN KINASE PIM-1
Common Name English
Code System Code Type Description
PHAROS
P11309
Created by admin on Tue Apr 01 16:59:35 GMT 2025 , Edited by admin on Tue Apr 01 16:59:35 GMT 2025
PRIMARY
FDA UNII
5NJ22TAB5Y
Created by admin on Tue Apr 01 16:59:35 GMT 2025 , Edited by admin on Tue Apr 01 16:59:35 GMT 2025
PRIMARY
CHEBI
87673
Created by admin on Tue Apr 01 16:59:35 GMT 2025 , Edited by admin on Tue Apr 01 16:59:35 GMT 2025
PRIMARY
UNIPROT
P11309
Created by admin on Tue Apr 01 16:59:35 GMT 2025 , Edited by admin on Tue Apr 01 16:59:35 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
Ki
INHIBITOR -> TARGET
COMPETITIVE INHIBITOR
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
COMPETITIVE INHIBITOR
Ki
INHIBITOR -> TARGET
Kd
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
PAN-PIM INHIBITOR
IC50
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_99] [1_189] [1_352] DEXFOSFOSERINE VI4F0K069V
AMINO ACID SUBSTITUTION [1_114] THREONINE PHOSPHATE 3L4WX7B1EI
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL