U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 16:55:42 GMT 2025
Edited
by admin
on Tue Apr 01 16:55:42 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
5M46696SR5
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CYCLIN-DEPENDENT KINASE 4
Common Name English
CELL DIVISION PROTEIN KINASE 4
Preferred Name English
CDK4
Common Name English
PSK-J3
Common Name English
Code System Code Type Description
PHAROS
P11802
Created by admin on Tue Apr 01 16:55:42 GMT 2025 , Edited by admin on Tue Apr 01 16:55:42 GMT 2025
PRIMARY
UNIPROT
P11802
Created by admin on Tue Apr 01 16:55:42 GMT 2025 , Edited by admin on Tue Apr 01 16:55:42 GMT 2025
PRIMARY
FDA UNII
5M46696SR5
Created by admin on Tue Apr 01 16:55:42 GMT 2025 , Edited by admin on Tue Apr 01 16:55:42 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Ki
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
WEAK INHIBITOR->TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IN-VITRO, IN-VIVO
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
WEAK INHIBITOR->TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
CELL-FREE KINASE ASSY (CDK4/CYCLIN D1)
INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
PRECLINICAL
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_1] N-ACETYLALANINE 26C4VY6Z0M
AMINO ACID SUBSTITUTION [1_171] THREONINE PHOSPHATE 3L4WX7B1EI
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL