U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:32:02 GMT 2025
Edited
by admin
on Tue Apr 01 18:32:02 GMT 2025
Protein Type RECEPTOR
Protein Sub Type G PROTEIN-COUPLED RECEPTOR
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
5CLY6W2H1M
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CORTICOTROPIN-RELEASING FACTOR RECEPTOR 1
Common Name English
CORTICOTROPIN RELEASING FACTOR SUBTYPE 1 RECEPTOR
Preferred Name English
CRFR-1
Common Name English
CRF-1
Common Name English
CRF1
Common Name English
Code System Code Type Description
FDA UNII
5CLY6W2H1M
Created by admin on Tue Apr 01 18:32:02 GMT 2025 , Edited by admin on Tue Apr 01 18:32:02 GMT 2025
PRIMARY
From To
1_7 1_31
1_21 1_64
1_45 1_79
1_194 1_264
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_15
N 1_22
N 1_55
N 1_67
N 1_75
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
Ki
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_307] SERINE DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL