U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 09:08:40 GMT 2025
Edited
by admin
on Wed Apr 02 09:08:40 GMT 2025
Protein Type ENZYME
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
57DB6RY8JM
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ATP-DEPENDENT HELICASE SMARCA2
Preferred Name English
PROBABLE GLOBAL TRANSCRIPTION ACTIVATOR SNF2L2
Common Name English
PROTEIN BRAHMA HOMOLOG
Common Name English
BAF190B
Common Name English
SWI/SNF-RELATED MATRIX-ASSOCIATED ACTIN-DEPENDENT REGULATOR OF CHROMATIN SUBFAMILY A MEMBER 2
Common Name English
SNF2-ALPHA
Common Name English
BRG1-ASSOCIATED FACTOR 190B
Common Name English
HBRM
Common Name English
Code System Code Type Description
FDA UNII
57DB6RY8JM
Created by admin on Wed Apr 02 09:08:40 GMT 2025 , Edited by admin on Wed Apr 02 09:08:40 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
Potently and selectively inhibits the ATPase components of the BAF complex, resulting in BAF Inhibition.
ALLOSTERIC INHIBITOR

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_190] [1_604] [1_997] [1_999] SITE_SPECIFIC N6-ACETYLLYSINE 470AD5VY1X
AMINO_ACID_SUBSTITUTION [1_172] [1_175] [1_316] [1_329] [1_588] [1_666] [1_670] [1_1377] [1_1512] [1_1516] [1_1528] [1_1568] [1_1572] SITE_SPECIFIC DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL