Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 16:34:19 GMT 2025
by
admin
on
Tue Apr 01 16:34:19 GMT 2025
|
| Protein Type | RECEPTOR |
| Protein Sub Type | |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
50U1BO5G5P
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
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Common Name | English | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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P08913
Created by
admin on Tue Apr 01 16:34:19 GMT 2025 , Edited by admin on Tue Apr 01 16:34:19 GMT 2025
|
PRIMARY | |||
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ALPHA-2_ADRENERGIC_RECEPTOR#INDIVIDUAL
Created by
admin on Tue Apr 01 16:34:19 GMT 2025 , Edited by admin on Tue Apr 01 16:34:19 GMT 2025
|
PRIMARY | |||
|
50U1BO5G5P
Created by
admin on Tue Apr 01 16:34:19 GMT 2025 , Edited by admin on Tue Apr 01 16:34:19 GMT 2025
|
PRIMARY | |||
|
P08913
Created by
admin on Tue Apr 01 16:34:19 GMT 2025 , Edited by admin on Tue Apr 01 16:34:19 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_106 | 1_188 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_10 |
| N | 1_14 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
|
AGONIST -> TARGET | |||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
INHIBITOR -> TARGET |
Ki
|
||
|
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
|
||
|
|
AGONIST -> TARGET | |||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
|
RADIOLIGAND->TARGET | |||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
|
AGONIST -> TARGET |
|
||
|
|
INHIBITOR -> TARGET |
At small doses, 1-PP (ED50 = 80 ?g/kg, i.v.) reversed the depressant effect of the ?2-adrenoceptor agonist, clonidine
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
ACTIVATOR -> TARGET |
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
INHIBITOR -> TARGET | |||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
LIGAND->OFF TARGET |
IC50
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
INHIBITOR -> TARGET |
Radioligand assay in human platelets
IC50
|
||
|
AGONIST -> TARGET |
Ki
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
Has 0.78 relative activity
EC50
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
||
|
AGONIST -> TARGET |
SHORT-ACTING
|
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_331] | DEXFOSFOSERINE | VI4F0K069V |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| Molecular Formula | CHEMICAL |
|
||||
| MOL_WEIGHT | CHEMICAL |
|