U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
This repository is under review for potential modification in compliance with Administration directives.

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 23:44:30 GMT 2025
Edited
by admin
on Tue Apr 01 23:44:30 GMT 2025
Protein Type RECEPTOR
Protein Sub Type TYROSINE KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
4ZX3AX8QGO
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CD-246 F1174L
Preferred Name English
ANAPLASTIC LYMPHOMA KINASE F1174L
Common Name English
ALK TYROSINE KINASE RECEPTOR F1174L
Systematic Name English
CD246 F1174L
Code English
ALK F1174L MUTANT
Common Name English
Code System Code Type Description
UNIPROT
Q9UM73
Created by admin on Tue Apr 01 23:44:30 GMT 2025 , Edited by admin on Tue Apr 01 23:44:30 GMT 2025
PRIMARY
WIKIPEDIA
ANAPLASTIC LYMPHOMA KINASE
Created by admin on Tue Apr 01 23:44:30 GMT 2025 , Edited by admin on Tue Apr 01 23:44:30 GMT 2025
PRIMARY
FDA UNII
4ZX3AX8QGO
Created by admin on Tue Apr 01 23:44:30 GMT 2025 , Edited by admin on Tue Apr 01 23:44:30 GMT 2025
PRIMARY
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_151
N 1_226
N 1_267
N 1_306
N 1_393
N 1_406
N 1_427
N 1_545
N 1_553
N 1_609
N 1_691
N 1_790
N 1_845
N 1_846
N 1_868
N 1_968
Related Record Type Details
INHIBITOR -> TARGET
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_1060] [1_1074] [1_1078] [1_1113] [1_1260] [1_1489] [1_1586] TYROSINE O-PHOSPHATE 2R86C98KDX
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL
Molecular Formula CHEMICAL