Details
| Stereochemistry | ABSOLUTE |
| Molecular Formula | C20H27NO2.ClH |
| Molecular Weight | 349.895 |
| Optical Activity | UNSPECIFIED |
| Defined Stereocenters | 3 / 3 |
| E/Z Centers | 0 |
| Charge | 0 |
SHOW SMILES / InChI
SMILES
Cl.OC1=CC2=C(C[C@H]3N(CC4CC4)CC[C@@]25CCCC[C@@]35O)C=C1
InChI
InChIKey=QWGXEENWLDBHTR-QGPGBOAMSA-N
InChI=1S/C20H27NO2.ClH/c22-16-6-5-15-11-18-20(23)8-2-1-7-19(20,17(15)12-16)9-10-21(18)13-14-3-4-14;/h5-6,12,14,18,22-23H,1-4,7-11,13H2;1H/t18-,19+,20-;/m1./s1
| Molecular Formula | ClH |
| Molecular Weight | 36.461 |
| Charge | 0 |
| Count |
|
| Stereochemistry | ACHIRAL |
| Additional Stereochemistry | No |
| Defined Stereocenters | 0 / 0 |
| E/Z Centers | 0 |
| Optical Activity | NONE |
| Molecular Formula | C20H27NO2 |
| Molecular Weight | 313.4339 |
| Charge | 0 |
| Count |
|
| Stereochemistry | ABSOLUTE |
| Additional Stereochemistry | No |
| Defined Stereocenters | 3 / 3 |
| E/Z Centers | 0 |
| Optical Activity | UNSPECIFIED |
Oxilorphan (also known as levo-BC-2605) was developed as a long-acting, narcotic antagonist that has agonist properties. Oxilorphan is a partial agonist at the kappa-opioid receptor and antagonist of the mu-opioid receptor. During clinical trials, oxilorphan had led to dysphoria, which combined with its hallucinogenic effects, serves to limit its clinical usefulness. As a result, many patients who experienced these side effects refused to take additional doses in clinical trials.
Approval Year
| Substance Class |
Chemical
Created
by
admin
on
Edited
Fri Dec 15 15:35:52 GMT 2023
by
admin
on
Fri Dec 15 15:35:52 GMT 2023
|
| Record UNII |
4IJ68MD32N
|
| Record Status |
Validated (UNII)
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| Record Version |
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-
Download
| Name | Type | Language | ||
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Common Name | English | ||
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Systematic Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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42281-48-1
Created by
admin on Fri Dec 15 15:35:52 GMT 2023 , Edited by admin on Fri Dec 15 15:35:52 GMT 2023
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PRIMARY | |||
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52305-98-3
Created by
admin on Fri Dec 15 15:35:52 GMT 2023 , Edited by admin on Fri Dec 15 15:35:52 GMT 2023
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ALTERNATIVE | |||
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21159630
Created by
admin on Fri Dec 15 15:35:52 GMT 2023 , Edited by admin on Fri Dec 15 15:35:52 GMT 2023
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PRIMARY | |||
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4IJ68MD32N
Created by
admin on Fri Dec 15 15:35:52 GMT 2023 , Edited by admin on Fri Dec 15 15:35:52 GMT 2023
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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PARENT -> SALT/SOLVATE |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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ACTIVE MOIETY |