U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS
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Approval Year

Substance Class Protein
Created
by admin
on Wed Apr 02 02:47:16 GMT 2025
Edited
by admin
on Wed Apr 02 02:47:16 GMT 2025
Protein Type RECEPTOR
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
438XLITDI3
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
NUCLEAR RECEPTOR SUBFAMILY 1 GROUP I MEMBER 3
Common Name English
CAR
Preferred Name English
CONSTITUTIVE ACTIVATOR OF RETINOID RESPONSE
Common Name English
NR1I3
Common Name English
CONSTITUTIVE ANDROSTANE RECEPTOR
Common Name English
ORPHAN NUCLEAR RECEPTOR MB67
Common Name English
CONSTITUTIVE ACTIVE RESPONSE
Common Name English
Code System Code Type Description
FDA UNII
438XLITDI3
Created by admin on Wed Apr 02 02:47:16 GMT 2025 , Edited by admin on Wed Apr 02 02:47:16 GMT 2025
PRIMARY
Related Record Type Details
AGONIST -> TARGET
INHIBITOR
EC50
ACTIVATOR -> TARGET
ACTIVATOR

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO_ACID_SUBSTITUTION [1_11] [1_14] [1_28] [1_31] SITE_SPECIFIC C4-TYPE ZINC FINGER C56TF4V7OP
AMINO ACID SUBSTITUTION [1_38] THREONINE PHOSPHATE 3L4WX7B1EI
AMINO_ACID_SUBSTITUTION [1_47] [1_53] [1_63] [1_66] SITE_SPECIFIC C4-TYPE ZINC FINGER C56TF4V7OP
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL