U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Unknown
139594
Substance Class Protein
Created
by admin
on Sat Dec 16 12:08:54 GMT 2023
Edited
by admin
on Sat Dec 16 12:08:54 GMT 2023
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
3T7136LE8K
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
ALPHA-1A ADRENERGIC RECEPTOR
Common Name English
Adrenergic α1A receptor
Common Name English
ADRA1C
Common Name English
ALPHA-1A ADRENOCEPTOR
Common Name English
Adrenergic α1A
Common Name English
Adrenergic α1A
Common Name English
ALPHA-1A ADRENORECEPTOR
Common Name English
Code System Code Type Description
FDA UNII
3T7136LE8K
Created by admin on Sat Dec 16 12:08:56 GMT 2023 , Edited by admin on Sat Dec 16 12:08:56 GMT 2023
PRIMARY
PHAROS
P35348
Created by admin on Sat Dec 16 12:08:56 GMT 2023 , Edited by admin on Sat Dec 16 12:08:56 GMT 2023
PRIMARY
UNIPROT
P35348
Created by admin on Sat Dec 16 12:08:56 GMT 2023 , Edited by admin on Sat Dec 16 12:08:56 GMT 2023
PRIMARY
WIKIPEDIA
ALPHA-1_ADRENERGIC_RECEPTOR
Created by admin on Sat Dec 16 12:08:56 GMT 2023 , Edited by admin on Sat Dec 16 12:08:56 GMT 2023
PRIMARY
From To
1_99 1_176
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_7
N 1_13
N 1_22
Related Record Type Details
Structure of LABETALOL
AGONIST -> TARGET
Structure of NAFTOPIDIL
INHIBITOR -> TARGET
Ki
Structure of RS-97078 FREE BASE
INHIBITOR -> TARGET
Structure of BENZPHETAMINE
AGONIST -> TARGET
Structure of SILODOSIN
INHIBITOR -> TARGET
Selectivity of silodosin determined in cloned human α1-adrenergic receptor (α1-AR) subtypes in cultured Chinese hamster ovary cells.Silodosin has greater affinity for the α1A-adrenergic receptor than for the α1B-adrenergic receptor (by a factor of 583), minimizing the propensity for blood pressure-related adverse effects mediated by α1B blockade.
Ki
Structure of XYLOMETAZOLINE
AGONIST -> TARGET
Structure of PSEUDOEPHEDRINE
AGONIST -> TARGET
Structure of TERAZOSIN
INHIBITOR -> TARGET
Structure of OXEDRINE
AGONIST -> TARGET
Structure of DROXIDOPA
AGONIST -> TARGET
Structure of MOXISYLYTE
AGONIST -> TARGET
Structure of APRACLONIDINE
AGONIST -> TARGET
Structure of AROTINOLOL
AGONIST -> TARGET
Structure of MIDODRINE
AGONIST -> TARGET
Structure of PHENTOLAMINE
AGONIST -> TARGET
Structure of RS-100975
INHIBITOR -> TARGET
Structure of CHLORPROMAZINE
INHIBITOR -> TARGET
Structure of Prazosin H-3
RADIOLIGAND->TARGET
BINDING
Kd
Structure of NIAPRAZINE
INHIBITOR -> TARGET
Ki
Structure of ETILEFRINE
AGONIST -> TARGET
Structure of PRAZOSIN
INHIBITOR -> TARGET
BINDING
IC50
Structure of 6-FLUORO-DMT
AGONIST -> TARGET
Structure of OXYMETHOLONE
AGONIST -> TARGET
Structure of PALIPERIDONE
INHIBITOR -> TARGET
INHIBITOR
Ki
Structure of LABETALOL
INHIBITOR -> TARGET
Ki
Structure of TETRAHYDROZOLINE
AGONIST -> TARGET
Structure of FIDUXOSIN
INHIBITOR -> TARGET
Structure of PHENYLEPHRINE
AGONIST -> TARGET
Structure of TAPRIZOSIN
INHIBITOR -> TARGET
Structure of RWJ-38063
INHIBITOR -> TARGET
Structure of CIRAZOLINE
AGONIST -> TARGET
Structure of INDORAMIN
AGONIST -> TARGET
Structure of NAPHAZOLINE
AGONIST -> TARGET
Structure of TOLAZOLINE
AGONIST -> TARGET
Structure of TIAMENIDINE
AGONIST -> TARGET
Structure of 4-METHOXYAMPHETAMINE
AGONIST -> TARGET
Structure of EPINEPHRINE
AGONIST -> TARGET
BINDING
IC50
Structure of ROLUPERIDONE
INHIBITOR -> TARGET
Structure of ADIMOLOL
INHIBITOR -> TARGET
Structure of ALFUZOSIN
INHIBITOR -> TARGET
Structure of METHOXAMINE
AGONIST -> TARGET
Structure of DAPIPRAZOLE
INHIBITOR -> TARGET
Structure of SHI-437 FREE BASE
INHIBITOR -> TARGET
Structure of NOREPINEPHRINE
AGONIST -> TARGET
Structure of DABUZALGRON
AGONIST -> TARGET
Structure of PHENDIMETRAZINE
AGONIST -> TARGET
Structure of TRIMAZOSIN
AGONIST -> TARGET
Structure of TRIFLUOPERAZINE
INHIBITOR -> TARGET
Structure of UPIDOSIN
INHIBITOR -> TARGET
Structure of OXYMETAZOLINE
AGONIST -> TARGET
Structure of WB-4101
INHIBITOR -> TARGET
BINDING
IC50
Structure of CUMI-101 C-11
RADIOLIGAND->TARGET
REPRESENTIVE ALPHA-1 ADRENERGIC RECEPTOR
Ki
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL
NIH
NCATS
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