Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Thu Jul 06 17:45:25 UTC 2023
by
admin
on
Thu Jul 06 17:45:25 UTC 2023
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Protein Sub Type | |
Sequence Origin | HUMAN |
Sequence Type | COMPLETE |
Record UNII |
3T7136LE8K
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Record Status |
Validated (UNII)
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Record Version |
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-
Download
Name | Type | Language | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
Code System | Code | Type | Description | ||
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3T7136LE8K
Created by
admin on Thu Jul 06 17:45:27 UTC 2023 , Edited by admin on Thu Jul 06 17:45:27 UTC 2023
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PRIMARY | |||
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P35348
Created by
admin on Thu Jul 06 17:45:27 UTC 2023 , Edited by admin on Thu Jul 06 17:45:27 UTC 2023
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PRIMARY | |||
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P35348
Created by
admin on Thu Jul 06 17:45:27 UTC 2023 , Edited by admin on Thu Jul 06 17:45:27 UTC 2023
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PRIMARY | |||
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ALPHA-1_ADRENERGIC_RECEPTOR
Created by
admin on Thu Jul 06 17:45:27 UTC 2023 , Edited by admin on Thu Jul 06 17:45:27 UTC 2023
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PRIMARY |
From | To |
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1_99 | 1_176 |
Glycosylation Type | HUMAN |
Glycosylation Link Type | Site |
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N | 1_7 |
N | 1_13 |
N | 1_22 |
Related Record | Type | Details | ||
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AGONIST -> TARGET | |||
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INHIBITOR -> TARGET |
Ki
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INHIBITOR -> TARGET |
Selectivity of silodosin determined in cloned human α1-adrenergic receptor (α1-AR) subtypes in cultured Chinese hamster ovary cells.Silodosin has greater affinity for the α1A-adrenergic receptor than for the α1B-adrenergic receptor (by a factor of 583), minimizing the propensity for blood pressure-related adverse effects mediated by α1B blockade.
Ki
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
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AGONIST -> TARGET | |||
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INHIBITOR -> TARGET |
INHIBITOR
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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INHIBITOR -> TARGET |
Ki
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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AGONIST -> TARGET |
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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RADIOLIGAND->TARGET |
REPRESENTIVE ALPHA-1 ADRENERGIC RECEPTOR
Ki
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Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
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MOL_WEIGHT | CHEMICAL |
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