Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Wed Apr 02 02:45:05 GMT 2025
by
admin
on
Wed Apr 02 02:45:05 GMT 2025
|
| Protein Type | ENZYME |
| Protein Sub Type | TYROSINE KINASE |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
3M5IJI39XM
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Preferred Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English | ||
|
Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
3M5IJI39XM
Created by
admin on Wed Apr 02 02:45:05 GMT 2025 , Edited by admin on Wed Apr 02 02:45:05 GMT 2025
|
PRIMARY |
| From | To |
|---|---|
| 1_4 | 1_31 |
| 1_131 | 1_161 |
| 1_164 | 1_172 |
| 1_168 | 1_180 |
| 1_188 | 1_196 |
| 1_192 | 1_204 |
| 1_205 | 1_213 |
| 1_209 | 1_221 |
| 1_224 | 1_233 |
| 1_237 | 1_264 |
| 1_268 | 1_279 |
| 1_283 | 1_298 |
| 1_301 | 1_305 |
| 1_478 | 1_487 |
| 1_482 | 1_495 |
| 1_498 | 1_507 |
| 1_511 | 1_527 |
| 1_530 | 1_544 |
| 1_534 | 1_552 |
| 1_555 | 1_564 |
| 1_568 | 1_589 |
| 1_592 | 1_600 |
| 1_596 | 1_608 |
| Glycosylation Type | HUMAN |
| Glycosylation Link Type | Site |
|---|---|
| N | 1_113 |
| N | 1_149 |
| N | 1_156 |
| N | 1_228 |
| N | 1_333 |
| N | 1_385 |
| N | 1_448 |
| N | 1_470 |
| N | 1_523 |
| N | 1_551 |
| N | 1_595 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
INHIBITOR->OFF-TARGET |
|
||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IC50
|
||
|
|
INHIBITOR -> TARGET | |||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
IRREVERSIBLE INHIBITOR
IC50
|
||
|
INHIBITOR -> TARGET |
IC50
|
||
|
|
INHIBITOR -> TARGET | |||
|
|
INHIBITOR -> TARGET | |||
|
INHIBITOR -> TARGET |
|
||
|
INHIBITOR -> TARGET |
Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO ACID SUBSTITUTION | [1_850] [1_1010] [1_1031] [1_1125] [1_1137] [1_1163] [1_1177] [1_1217] [1_1233] [1_1259] | TYROSINE O-PHOSPHATE | 2R86C98KDX |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
|