U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Mon Mar 31 23:17:22 GMT 2025
Edited
by admin
on Mon Mar 31 23:17:22 GMT 2025
Protein Type MONOCLONAL ANTIBODY CONJUGATE
Protein Sub Type IGG1
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
3F0FR4W3H8
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
INDUSATUMAB VEDOTIN
INN   WHO-DD  
INN  
Official Name English
MLN-0264
Preferred Name English
Indusatumab vedotin [WHO-DD]
Common Name English
TAK-264
Code English
MLN0264
Code English
RECOMBINANT HUMAN IgG1 KAPPA ANTI-GUANYL CYCLASE C MONOCLONAL ANTIBODY MLN2045 - MONOMETHYL AURISTATIN E CONJUGATE
Common Name English
indusatumab vedotin [INN]
Common Name English
Classification Tree Code System Code
FDA ORPHAN DRUG 437914
Created by admin on Mon Mar 31 23:17:22 GMT 2025 , Edited by admin on Mon Mar 31 23:17:22 GMT 2025
FDA ORPHAN DRUG 438014
Created by admin on Mon Mar 31 23:17:22 GMT 2025 , Edited by admin on Mon Mar 31 23:17:22 GMT 2025
Code System Code Type Description
FDA UNII
3F0FR4W3H8
Created by admin on Mon Mar 31 23:17:22 GMT 2025 , Edited by admin on Mon Mar 31 23:17:22 GMT 2025
PRIMARY
NCI_THESAURUS
C101524
Created by admin on Mon Mar 31 23:17:22 GMT 2025 , Edited by admin on Mon Mar 31 23:17:22 GMT 2025
PRIMARY
CAS
1514889-12-3
Created by admin on Mon Mar 31 23:17:22 GMT 2025 , Edited by admin on Mon Mar 31 23:17:22 GMT 2025
PRIMARY
DRUG BANK
DB12413
Created by admin on Mon Mar 31 23:17:22 GMT 2025 , Edited by admin on Mon Mar 31 23:17:22 GMT 2025
PRIMARY
INN
10033
Created by admin on Mon Mar 31 23:17:22 GMT 2025 , Edited by admin on Mon Mar 31 23:17:22 GMT 2025
PRIMARY
WIKIPEDIA
Indusatumab vedotin
Created by admin on Mon Mar 31 23:17:22 GMT 2025 , Edited by admin on Mon Mar 31 23:17:22 GMT 2025
PRIMARY
SMS_ID
300000025303
Created by admin on Mon Mar 31 23:17:22 GMT 2025 , Edited by admin on Mon Mar 31 23:17:22 GMT 2025
PRIMARY
From To
1_22 1_95
1_146 1_202
1_263 1_323
1_369 1_427
2_22 2_95
2_146 2_202
2_263 2_323
2_369 2_427
3_23 3_88
3_134 3_194
4_23 4_88
4_134 4_194
1_222 3_214
2_222 4_214
1_228 2_228
1_231 2_231
Glycosylation Type MAMMALIAN
Glycosylation Link Type Site
N 1_299
N 2_299
Related Record Type Details
PARENT -> CONJUGATE
TARGET->CONJUGATED TOXIN
Related Record Type Details
ACTIVE MOIETY

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_222] [1_228] [1_231] [2_222] [2_228] [2_231] [3_214] [4_214] C Amount: Cysteinyl vedotin 6603L01WUR
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT:NUMBER(CALCULATED) CHEMICAL