Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 16:33:23 GMT 2025
by
admin
on
Tue Apr 01 16:33:23 GMT 2025
|
| Protein Type | ENZYME |
| Protein Sub Type | CYTOCHROME P450 |
| Sequence Origin | HUMAN |
| Sequence Type | COMPLETE |
| Record UNII |
31I8UTYA8X
|
| Record Status |
Validated (UNII)
|
| Record Version |
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-
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| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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31I8UTYA8X
Created by
admin on Tue Apr 01 16:33:23 GMT 2025 , Edited by admin on Tue Apr 01 16:33:23 GMT 2025
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PRIMARY | |||
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P19099
Created by
admin on Tue Apr 01 16:33:23 GMT 2025 , Edited by admin on Tue Apr 01 16:33:23 GMT 2025
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PRIMARY | |||
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P19099
Created by
admin on Tue Apr 01 16:33:23 GMT 2025 , Edited by admin on Tue Apr 01 16:33:23 GMT 2025
|
PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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SUBSTRATE -> METABOLIC ENZYME | |||
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INHIBITOR -> TARGET |
Shows selectivity for CYP11B2 over CYP11B1.
IC50
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RADIOLIGAND->TARGET |
No selectivity for CYP11B2 over CYP11B1.
IC50
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET |
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INHIBITOR -> TARGET | |||
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RADIOLIGAND->TARGET |
Selectivity for CYP11B2 over CYP11B1 was higher for CDP2230 than for MTO and IMTO.
IC50
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INHIBITOR -> TARGET |
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TISSUE EXPRESSION -> PARENT |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT | CHEMICAL |
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