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Details

Stereochemistry ABSOLUTE
Molecular Formula C32H30F9N4O5.K
Molecular Weight 760.6883
Optical Activity UNSPECIFIED
Defined Stereocenters 2 / 2
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of Obicetrapib potassium

SMILES

[K+].CCOC(=O)N1[C@H](CC)C[C@H](N(CC2=CC(=CC(=C2)C(F)(F)F)C(F)(F)F)C3=NC=C(OCCCC([O-])=O)C=N3)C4=C1C=CC(=C4)C(F)(F)F

InChI

InChIKey=GEUMGSDQIGYWML-IINJVQNMSA-M
InChI=1S/C32H31F9N4O5.K/c1-3-22-14-26(24-13-19(30(33,34)35)7-8-25(24)45(22)29(48)49-4-2)44(28-42-15-23(16-43-28)50-9-5-6-27(46)47)17-18-10-20(31(36,37)38)12-21(11-18)32(39,40)41;/h7-8,10-13,15-16,22,26H,3-6,9,14,17H2,1-2H3,(H,46,47);/q;+1/p-1/t22-,26+;/m1./s1

HIDE SMILES / InChI

Molecular Formula C32H30F9N4O5
Molecular Weight 721.59
Charge -1
Count
Stereochemistry ABSOLUTE
Additional Stereochemistry No
Defined Stereocenters 2 / 2
E/Z Centers 0
Optical Activity UNSPECIFIED

Molecular Formula K
Molecular Weight 39.0983
Charge 1
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Approval Year

Substance Class Chemical
Created
by admin
on Tue Apr 01 18:59:19 GMT 2025
Edited
by admin
on Tue Apr 01 18:59:19 GMT 2025
Record UNII
2PBJ8V9F6I
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
Obicetrapib potassium
Common Name English
(2R,4S)-4-[[3,5-Bis(trifluoromethyl)benzyl][5-(3-carboxypropoxy)pyrimidin-2-yl]amino]-2-ethyl-6-trifluoromethyl-3,4-dihydro-2H-quinoline-1-carboxylic acid ethyl ester potassium salt
Preferred Name English
1(2H)-Quinolinecarboxylic acid, 4-[[[3,5-bis(trifluoromethyl)phenyl]methyl][5-(3-carboxypropoxy)-2-pyrimidinyl]amino]-2-ethyl-3,4-dihydro-6-(trifluoromethyl)-, 1-ethyl ester, potassium salt (1:1), (2R,4S)-
Systematic Name English
Code System Code Type Description
CAS
866399-90-8
Created by admin on Tue Apr 01 18:59:19 GMT 2025 , Edited by admin on Tue Apr 01 18:59:19 GMT 2025
PRIMARY
SMS_ID
300000013045
Created by admin on Tue Apr 01 18:59:19 GMT 2025 , Edited by admin on Tue Apr 01 18:59:19 GMT 2025
PRIMARY
PUBCHEM
121596646
Created by admin on Tue Apr 01 18:59:19 GMT 2025 , Edited by admin on Tue Apr 01 18:59:19 GMT 2025
PRIMARY
FDA UNII
2PBJ8V9F6I
Created by admin on Tue Apr 01 18:59:19 GMT 2025 , Edited by admin on Tue Apr 01 18:59:19 GMT 2025
PRIMARY
Related Record Type Details
PARENT -> SALT/SOLVATE
Related Record Type Details
ACTIVE MOIETY