Cyprodime

COC1=C2C(C[C@H]3N(CC4CC4)CC[C@@]25CC(=O)CC[C@@]35OC)=CC=C1

InChIKey=INUCRGMCKDQKNA-CEMLEFRQSA-N

InChI=1S/C22H29NO3/c1-25-18-5-3-4-16-12-19-22(26-2)9-8-17(24)13-21(22,20(16)18)10-11-23(19)14-15-6-7-15/h3-5,15,19H,6-14H2,1-2H3/t19-,21-,22-/m1/s1

Stereochemistry	ABSOLUTE
Additional Stereochemistry	No
Defined Stereocenters	3 / 3
E/Z Centers	0
Optical Activity	UNSPECIFIED

Targets

Primary Target	Pharmacology	Condition	Potency
Mu-type opioid receptor 61 Target ID: P33535\|\|\|Q64064 Gene ID: 25601.0 Gene Symbol: Oprm1 Target Organism: Rattus norvegicus (Rat) Sources: https://www.ncbi.nlm.nih.gov/pubmed/2536439	Antagonist 2849		5.4 nM [Ki]

Substance Class	Chemical Created by `admin` on `Mon Mar 31 22:54:12 GMT 2025` Edited by `admin` on `Mon Mar 31 22:54:12 GMT 2025`
Record UNII	2C6F5L8S8X
Record Status	`Validated (UNII)`
Record Version

Name

Type

Language

(4bR,8aR,9R)-11-(cyclopropylmethyl)-4,8a-dimethoxy-8,8a,9,10-tetrahydro-5H-9,4b-(epiminoethano)phenanthren-6(7H)-one hydrochloride

Preferred Name

English

Cyprodime

Common Name

English

MORPHINAN-6-ONE, 17-(CYCLOPROPYLMETHYL)-4,14-DIMETHOXY-

Systematic Name

English

17-(Cyclopropylmethyl)-4,14-dimethoxymorphinan-6-one

Systematic Name

English

Code System Code Type Description

CAS

118111-54-9