U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sun Dec 18 09:07:56 UTC 2022
Edited
by admin
on Sun Dec 18 09:07:56 UTC 2022
Protein Sub Type
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
2BJ58BX78W
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
KAPPA-TYPE OPIOID RECEPTOR
Common Name English
OPRK1
Common Name English
OPRK
Common Name English
K-OR-1
Common Name English
Code System Code Type Description
FDA UNII
2BJ58BX78W
Created by admin on Sun Dec 18 09:07:59 UTC 2022 , Edited by admin on Sun Dec 18 09:07:59 UTC 2022
PRIMARY
From To
1_131 1_210
Glycosylation Type HUMAN
Glycosylation Link Type Site
N 1_25
N 1_39
Related Record Type Details
AGONIST -> TARGET
PARTIAL AGONIST->TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
Ki
INHIBITOR -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
IC50
RADIOLIGAND->TARGET
Ki
RADIOLIGAND->TARGET
NON-INHIBITOR->OFF TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
Selective for the kappa receptor no mu activity.
RADIOLIGAND->TARGET
Ki
AGONIST -> TARGET
AGONIST -> TARGET
IC50
AGONIST -> TARGET
AGONIST -> TARGET
PARTIAL AGONIST->TARGET
INHIBITOR -> TARGET
RADIOLIGAND->TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
BINDING
Ki
INHIBITOR -> TARGET
AGONIST -> TARGET
NON-INHIBITOR->OFF TARGET
AGONIST -> TARGET
TARGET -> AGONIST
AGONIST -> TARGET
LIGAND->TARGET
TARGET->RADIOLIGAND
Ki
TARGET->RADIOLIGAND
Ki
INHIBITOR -> TARGET
ANTAGONIST
INHIBITOR -> TARGET
AGONIST -> TARGET
AGONIST -> TARGET
RADIOLIGAND->TARGET
Ki
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL