Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Sun Dec 18 09:07:56 UTC 2022
by
admin
on
Sun Dec 18 09:07:56 UTC 2022
|
Protein Sub Type | |
Sequence Origin | HUMAN |
Sequence Type | COMPLETE |
Record UNII |
2BJ58BX78W
|
Record Status |
Validated (UNII)
|
Record Version |
|
-
Download
Name | Type | Language | ||
---|---|---|---|---|
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
Code System | Code | Type | Description | ||
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2BJ58BX78W
Created by
admin on Sun Dec 18 09:07:59 UTC 2022 , Edited by admin on Sun Dec 18 09:07:59 UTC 2022
|
PRIMARY |
From | To |
---|---|
1_131 | 1_210 |
Glycosylation Type | HUMAN |
Glycosylation Link Type | Site |
---|---|
N | 1_25 |
N | 1_39 |
Related Record | Type | Details | ||
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AGONIST -> TARGET | |||
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PARTIAL AGONIST->TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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AGONIST -> TARGET |
Ki
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET | |||
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AGONIST -> TARGET | |||
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INHIBITOR -> TARGET |
IC50
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RADIOLIGAND->TARGET |
Ki
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RADIOLIGAND->TARGET | |||
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NON-INHIBITOR->OFF TARGET |
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AGONIST -> TARGET | |||
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET | |||
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AGONIST -> TARGET |
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INHIBITOR -> TARGET |
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AGONIST -> TARGET |
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AGONIST -> TARGET |
Selective for the kappa receptor no mu activity.
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RADIOLIGAND->TARGET |
Ki
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AGONIST -> TARGET |
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AGONIST -> TARGET |
IC50
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AGONIST -> TARGET | |||
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AGONIST -> TARGET | |||
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PARTIAL AGONIST->TARGET | |||
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INHIBITOR -> TARGET | |||
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RADIOLIGAND->TARGET | |||
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INHIBITOR -> TARGET | |||
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INHIBITOR -> TARGET |
BINDING
Ki
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INHIBITOR -> TARGET | |||
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AGONIST -> TARGET | |||
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NON-INHIBITOR->OFF TARGET |
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AGONIST -> TARGET | |||
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TARGET -> AGONIST | |||
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AGONIST -> TARGET |
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LIGAND->TARGET | |||
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TARGET->RADIOLIGAND |
Ki
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TARGET->RADIOLIGAND |
Ki
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INHIBITOR -> TARGET |
ANTAGONIST
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INHIBITOR -> TARGET | |||
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AGONIST -> TARGET |
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AGONIST -> TARGET |
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RADIOLIGAND->TARGET |
Ki
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Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
---|---|---|---|---|---|---|
MOL_WEIGHT | CHEMICAL |
|