U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 08:18:01 UTC 2023
Edited
by admin
on Sat Dec 16 08:18:01 UTC 2023
Protein Type MONOCLONAL ANTIBODY
Protein Sub Type IGG1
Sequence Origin HUMANIZED MOUSE
Sequence Type COMPLETE
Record UNII
237GB6IDKO
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
TIGATUZUMAB
INN   WHO-DD  
INN  
Official Name English
ANTI-TRAIL-R2 MOAB
Common Name English
Tigatuzumab [WHO-DD]
Common Name English
CS-1008
Code English
IMMUNOGLOBULIN G1, ANTI-(HUMAN CYTOKINE RECEPTOR DR5 (DEATH RECEPTOR 5)) (HUMAN-MOUSE MONOCLONAL TRA-8 .GAMMA.1-CHAIN), DISULFIDE WITH HUMAN-MOUSE MONOCLONAL TRA-8 .KAPPA.-CHAIN, DIMER
Systematic Name English
ANTI-DR5 MOAB
Common Name English
tigatuzumab [INN]
Common Name English
TRA-8
Code English
Classification Tree Code System Code
NCI_THESAURUS C20401
Created by admin on Sat Dec 16 08:18:01 UTC 2023 , Edited by admin on Sat Dec 16 08:18:01 UTC 2023
Code System Code Type Description
INN
8979
Created by admin on Sat Dec 16 08:18:01 UTC 2023 , Edited by admin on Sat Dec 16 08:18:01 UTC 2023
PRIMARY
FDA UNII
237GB6IDKO
Created by admin on Sat Dec 16 08:18:01 UTC 2023 , Edited by admin on Sat Dec 16 08:18:01 UTC 2023
PRIMARY
WIKIPEDIA
TIGATUZUMAB
Created by admin on Sat Dec 16 08:18:01 UTC 2023 , Edited by admin on Sat Dec 16 08:18:01 UTC 2023
PRIMARY
DRUG BANK
DB15101
Created by admin on Sat Dec 16 08:18:01 UTC 2023 , Edited by admin on Sat Dec 16 08:18:01 UTC 2023
PRIMARY
NCI_THESAURUS
C62482
Created by admin on Sat Dec 16 08:18:01 UTC 2023 , Edited by admin on Sat Dec 16 08:18:01 UTC 2023
PRIMARY
EVMPD
SUB124908
Created by admin on Sat Dec 16 08:18:01 UTC 2023 , Edited by admin on Sat Dec 16 08:18:01 UTC 2023
PRIMARY
ChEMBL
CHEMBL1743080
Created by admin on Sat Dec 16 08:18:01 UTC 2023 , Edited by admin on Sat Dec 16 08:18:01 UTC 2023
PRIMARY
CAS
918127-53-4
Created by admin on Sat Dec 16 08:18:01 UTC 2023 , Edited by admin on Sat Dec 16 08:18:01 UTC 2023
PRIMARY
From To
1_22 1_96
1_146 1_202
1_222 3_213
1_228 2_228
1_231 2_231
1_263 1_323
1_369 1_427
2_22 2_96
2_146 2_202
2_222 4_213
2_263 2_323
2_369 2_427
3_23 3_88
3_133 3_193
4_23 4_88
4_133 4_193
Glycosylation Type MAMMALIAN
Glycosylation Link Type Site
N 1_299
N 2_299
Related Record Type Details
TARGET -> INHIBITOR
Related Record Type Details
ACTIVE MOIETY
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT:ESTIMATE CHEMICAL
Molecular Formula CHEMICAL