U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 17:39:29 GMT 2025
Edited
by admin
on Tue Apr 01 17:39:29 GMT 2025
Protein Sub Type
Sequence Type COMPLETE
Record UNII
1GK9YLL8E0
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CAMP-SPECIFIC 3',5'-CYCLIC PHOSPHODIESTERASE 4B
Common Name English
DPDE4
Preferred Name English
PDE4B
Common Name English
PDE32
Common Name English
Code System Code Type Description
FDA UNII
1GK9YLL8E0
Created by admin on Tue Apr 01 17:39:29 GMT 2025 , Edited by admin on Tue Apr 01 17:39:29 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
RADIOLIGAND->TARGET
Good selectivity over PDE4D, excellent brain permeability, and a high level of specific binding in the “cold tracer” study.
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET
IC50
INHIBITOR -> TARGET

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_290] [1_659] [1_661] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL