Approval Year
Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 19:55:25 GMT 2025
by
admin
on
Tue Apr 01 19:55:25 GMT 2025
|
Protein Sub Type | |
Sequence Type | COMPLETE |
Record UNII |
11F03GK3UH
|
Record Status |
Validated (UNII)
|
Record Version |
|
-
Download
Name | Type | Language | ||
---|---|---|---|---|
|
Common Name | English | ||
|
Preferred Name | English | ||
|
Common Name | English |
Classification Tree | Code System | Code | ||
---|---|---|---|---|
|
CFR |
21 CFR 862.1650
Created by
admin on Tue Apr 01 19:55:25 GMT 2025 , Edited by admin on Tue Apr 01 19:55:25 GMT 2025
|
Code System | Code | Type | Description | ||
---|---|---|---|---|---|
|
625326-52-5
Created by
admin on Tue Apr 01 19:55:25 GMT 2025 , Edited by admin on Tue Apr 01 19:55:25 GMT 2025
|
ALTERNATIVE | |||
|
PKLR
Created by
admin on Tue Apr 01 19:55:25 GMT 2025 , Edited by admin on Tue Apr 01 19:55:25 GMT 2025
|
PRIMARY | |||
|
EC 2.7.1.40
Created by
admin on Tue Apr 01 19:55:25 GMT 2025 , Edited by admin on Tue Apr 01 19:55:25 GMT 2025
|
PRIMARY | |||
|
479853-13-9
Created by
admin on Tue Apr 01 19:55:25 GMT 2025 , Edited by admin on Tue Apr 01 19:55:25 GMT 2025
|
PRIMARY | |||
|
P30613
Created by
admin on Tue Apr 01 19:55:25 GMT 2025 , Edited by admin on Tue Apr 01 19:55:25 GMT 2025
|
PRIMARY | |||
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391970-89-1
Created by
admin on Tue Apr 01 19:55:25 GMT 2025 , Edited by admin on Tue Apr 01 19:55:25 GMT 2025
|
ALTERNATIVE | |||
|
11F03GK3UH
Created by
admin on Tue Apr 01 19:55:25 GMT 2025 , Edited by admin on Tue Apr 01 19:55:25 GMT 2025
|
PRIMARY |
Related Record | Type | Details | ||
---|---|---|---|---|
|
ACTIVATOR -> TARGET |
EC50
|
||
|
ACTIVATOR -> TARGET |
activator to 89% of activity
EC50
|
||
|
ACTIVATOR -> TARGET |
519% activation over baseline
ALLOSTERIC
EC50
|
Structural Modifications
Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
---|---|---|---|---|---|---|
AMINO ACID REPLACEMENT | [1_148] [2_418] [3_418] [4_418] | TYROSINE | TYROSINE O-PHOSPHATE | 2R86C98KDX | ||
AMINO ACID REPLACEMENT | [1_105] [1_313] [1_365] [2_105] [2_313] [2_365] [3_105] [3_313] [3_365] [4_105] [4_313] [4_365] | LYSINE | N6-SUCCINYLLYSINE | 3LH35AJA5L | ||
AMINO ACID REPLACEMENT | [1_2] [1_19] [1_26] [1_43] [1_140] [1_292] [2_2] [2_19] [2_26] [2_43] [2_140] [2_292] [3_2] [3_19] [3_26] [3_43] [3_140] [3_292] [4_2] [4_19] [4_26] [4_43] [4_140] [4_292] | SERINE | DEXFOSFOSERINE | VI4F0K069V | ||
AMINO ACID REPLACEMENT | [1_109] [1_365] [1_541] [2_109] [2_365] [2_541] [3_109] [3_365] [3_541] [4_109] [4_365] [4_541] | LYSINE | N6-SUCCINYLLYSINE | 3LH35AJA5L |
Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
---|---|---|---|---|---|---|
MOL_WEIGHT:NUMBER AVERAGE(CALCULATED) | CHEMICAL |
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Molecular Formula | CHEMICAL |
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