U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Sat Dec 16 12:23:24 UTC 2023
Edited
by admin
on Sat Dec 16 12:23:24 UTC 2023
Protein Sub Type
Sequence Type COMPLETE
Record UNII
0JQ7O17JE9
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
RHO-ASSOCIATED PROTEIN KINASE 2
Common Name English
RHO-ASSOCIATED, COILED-COIL-CONTAINING PROTEIN KINASE II
Common Name English
ROCK-II
Common Name English
RHO-ASSOCIATED, COILED-COIL-CONTAINING PROTEIN KINASE 2
Common Name English
KIAA0619
Common Name English
RHO KINASE 2
Common Name English
ROCK2
Common Name English
P164 ROCK-2
Common Name English
Code System Code Type Description
FDA UNII
0JQ7O17JE9
Created by admin on Sat Dec 16 12:23:25 UTC 2023 , Edited by admin on Sat Dec 16 12:23:25 UTC 2023
PRIMARY
UNIPROT
O75116
Created by admin on Sat Dec 16 12:23:25 UTC 2023 , Edited by admin on Sat Dec 16 12:23:25 UTC 2023
PRIMARY
PHAROS
O75116
Created by admin on Sat Dec 16 12:23:25 UTC 2023 , Edited by admin on Sat Dec 16 12:23:25 UTC 2023
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
ROCK2 selective inhibitor
INHIBITOR -> TARGET
INHIBITION OF THE PHOSPHORYLTRANSFERASE ACTIVITY OF THE KINASE
INHIBITOR
Ki
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITION OF THE PHOSPHORYLTRANSFERASE ACTIVITY OF THE KINASE
INHIBITOR
Ki
INHIBITOR -> TARGET
INHIBITOR -> TARGET
COMPETITIVE INHIBITOR
IC50
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
INHIBITOR -> TARGET
Inhibits signal transducer and activator of transcription 3 (STAT3) phosphorylation. Shifts T helper 17 (Th17)/T regulatory (Treg) balance towards the Treg phenotype
IC50
INHIBITOR -> TARGET
Competitive for ATP
Ki
Name Property Type Amount Referenced Substance Defining Parameters References
MOL_WEIGHT CHEMICAL