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Details

Stereochemistry ACHIRAL
Molecular Formula C8H6S
Molecular Weight 134.198
Optical Activity NONE
Defined Stereocenters 0 / 0
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of THIANAPHTHENE

SMILES

S1C=CC2=C1C=CC=C2

InChI

InChIKey=FCEHBMOGCRZNNI-UHFFFAOYSA-N
InChI=1S/C8H6S/c1-2-4-8-7(3-1)5-6-9-8/h1-6H

HIDE SMILES / InChI

Molecular Formula C8H6S
Molecular Weight 134.198
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

Approval Year

PubMed

PubMed

TitleDatePubMed
Synthesis and biological activity of alpha-bromoacryloyl lexitropsin conjugates.
2005-11
Biodesulfurization of dibenzothiophene and other organic sulfur compounds by a newly isolated Microbacterium strain ZD-M2.
2005-06-01
Prediction of genotoxicity of chemical compounds by statistical learning methods.
2005-06
Hydroxylation activity of P450 BM-3 mutant F87V towards aromatic compounds and its application to the synthesis of hydroquinone derivatives from phenolic compounds.
2005-06
Triplet-triplet energy transfer controlled by the donor-acceptor distance in rigidly held palladium-containing cofacial bisporphyrins.
2005-05-20
Selective adsorption of thiophene and 1-benzothiophene on metal-ion-exchanged zeolites in organic medium.
2005-05-15
Efficient access to 2-aryl-3-substituted benzo[b]thiophenes.
2005-04-29
Synthesis and binding affinities of novel SRIF-mimicking beta-D-glucosides satisfying the requirement for a pi-cloud at C1.
2005-03-17
Poly(thiaheterohelicene): a stiff conjugated helical polymer comprised of fused benzothiophene rings.
2005-03-03
Benzothiophenes containing a piperazine side chain as selective ligands for the estrogen receptor alpha and their bioactivities in vivo.
2005-03-01
Desulfurization of dibenzothiophene, benzothiophene, and other thiophene analogs by a newly isolated bacterium, Gordonia alkanivorans strain 1B.
2005-03
In vitro metabolic fate of a novel structural class: evidence for the formation of a reactive intermediate on a benzothiophene moiety.
2005-02-28
Benzo[b]thiophenesulphonamide 1,1-dioxide derivatives inhibit tNOX activity in a redox state-dependent manner.
2005-02-28
Design, synthesis, and biological evaluation of novel potent and selective alphavbeta3/alphavbeta5 integrin dual inhibitors with improved bioavailability. Selection of the molecular core.
2005-02-24
Simultaneous determination of NSO-heterocycles, homocycles and their metabolites in groundwater of tar oil contaminated sites using LC with diode array UV and fluorescence detection.
2005-02-18
Organoboron compounds with an 8-hydroxyquinolato chelate and its derivatives: substituent effects on structures and luminescence.
2005-02-07
Thermophilic biodesulfurization of various heterocyclic sulfur compounds and crude straight-run light gas oil fraction by a newly isolated strain Mycobacterium phlei WU-0103.
2005-02
Endocrinology and hormone therapy in breast cancer: selective oestrogen receptor modulators and downregulators for breast cancer - have they lost their way?
2005
Adsorption, desorption, and conversion of thiophene on H-ZSM5.
2004-12-07
Screening of antimicrobial activity of diarylamines in the 2,3,5-trimethylbenzo[b]thiophene series: a structure-activity evaluation study.
2004-12-06
Synthesis and NMR spectroscopic studies of allylsulfanyl-N1-alkyl-N4-phenyl-1,4-phenylenediamines and their cyclization products, 2,3-dihydro-1-benzothiophenes and thiochromans.
2004-12
NH2-SEP-PAK cartridges for enrichment of Aromatic Sulfur Compounds from sea water: determination by GC-FID and GC-MS.
2004-10-28
Palladium-catalyzed tandem reaction of yne-propargylic carbonates with boronic acids: a simple method for the synthesis of fused aromatic rings through allene-mediated electrocyclization.
2004-10-25
Benzothiophene and naphthalene derived constrained SERMs.
2004-10-18
New 3-[4-(2,3-dihydro-14-benzodioxin-5-yl)piperazin-1-yl]-1-(5-substituted benzo[b]thiophen-3-yl)propanol derivatives with dual action at 5-HT(1A) serotonin receptors and serotonin transporter as a new class of antidepressants.
2004-07
Phenylpiperazinylmethylheterocycle derivatives: synthesis and dopamine receptor binding profiles.
2004-07
C17,20-lyase inhibitors I. Structure-based de novo design and SAR study of C17,20-lyase inhibitors.
2004-05-01
[Determination of sulfur compounds in fluid catalytic cracking gasoline by gas chromatography with a sulfur chemiluminescence detector].
2004-05
Synthesis and serotonergic activity of variously substituted (3-amido)phenylpiperazine derivatives and benzothiophene-4-piperazine derivatives: novel antagonists for the vascular 5-HT1B receptor.
2004-04
Design, synthesis and structure-activity relationship of novel RXR-selective modulators.
2004-03-22
Discovery of novel heteroaryl-substituted chalcones as inhibitors of TNF-alpha-induced VCAM-1 expression.
2004-03-22
Efficient isomer-pure synthesis of a benzo[b]thiophene analogue of pentacene.
2004-03-19
Synthesis and cytotoxic activity of lipophilic sulphonamide derivatives of the benzo[b]thiophene 1,1-dioxide.
2004-03-01
Synthesis of new thiophene and benzo[b]thiophene hydrazide derivatives as human NPY Y(5) antagonists.
2004-02-09
A synthesis of heteroaromatic analogues of 1-methyl-1,2,3,4-tetrahydroisoquinoline using the Pummerer-type cyclization reaction: observation of tandem cyclization reaction.
2004-02
Elimination of sulfur from aromatic heterocycles by a water-soluble arene ruthenium cluster: synthesis and molecular structure of [H2S2Ru4(C6H6)4]Cl2.
2004-01-21
Modulation of selective serotonin reuptake inhibitor and 5-HT1A antagonist activity in 8-aza-bicyclo[3.2.1]octane derivatives of 2,3-dihydro-1,4-benzodioxane.
2004-01-19
Combined application of stable carbon isotope analysis and specific metabolites determination for assessing in situ degradation of aromatic hydrocarbons in a tar oil-contaminated aquifer.
2004-01-15
Potent inhibition of human liver aldehyde oxidase by raloxifene.
2004-01
Monitoring toxicity of industrial wastewater and specific chemicals to a green alga, nitrifying bacteria and an aquatic bacterium.
2004
Advances in estrogen receptor biology: prospects for improvements in targeted breast cancer therapy.
2004
Structure-activity relationship of benzo[b]thiophene-2-sulfonamide derivatives as novel human chymase inhibitors.
2003-11-17
Reactions that generate aromatic molecules: is aromatic stabilization less or more advanced than bond changes at the transition state? Kinetic and thermodynamic acidities of rhenium carbene complexes.
2003-10-08
Nitrosation, nitration, and autoxidation of the selective estrogen receptor modulator raloxifene by nitric oxide, peroxynitrite, and reactive nitrogen/oxygen species.
2003-10
2,6-disubstituted pyran-4-one and thiopyran-4-one inhibitors of DNA-Dependent protein kinase (DNA-PK).
2003-09-15
Synthesis and binding affinities of fluoroalkylated raloxifenes.
2003-08-15
Target specificity of selective estrogen receptor modulators within human endometrial cancer cells.
2003-07
Selective estrogen receptor modulators.
2003-05
Design, synthesis and in vitro evaluation of novel benzo[b]thiophene derivatives as serotonin N-acetyltransferase (AANAT) inhibitors.
2003-04
Advances in breast cancer treatment and prevention: preclinical studies on aromatase inhibitors and new selective estrogen receptor modulators (SERMs).
2003
Patents
Substance Class Chemical
Created
by admin
on Mon Mar 31 19:29:19 GMT 2025
Edited
by admin
on Mon Mar 31 19:29:19 GMT 2025
Record UNII
073790YQ2G
Record Status Validated (UNII)
Record Version
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Name Type Language
THIANAPHTHENE
MI  
Common Name English
NSC-47196
Preferred Name English
THIANAPHTHENE [MI]
Common Name English
BENZOTHIOPHENE
Systematic Name English
BENZOTHIOFURAN
Common Name English
BENZO(B)THIOPHENE
Systematic Name English
Code System Code Type Description
CHEBI
35858
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY
MERCK INDEX
m10725
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY Merck Index
PUBCHEM
7221
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY
ECHA (EC/EINECS)
202-395-7
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY
CAS
11095-43-5
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
SUPERSEDED
CHEBI
35857
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY
CAS
95-15-8
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY
FDA UNII
073790YQ2G
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY
MESH
C088015
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY
WIKIPEDIA
Benzothiophene
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY
EPA CompTox
DTXSID2052736
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY
NSC
47196
Created by admin on Mon Mar 31 19:29:19 GMT 2025 , Edited by admin on Mon Mar 31 19:29:19 GMT 2025
PRIMARY