Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Tue Apr 01 19:40:57 GMT 2025
by
admin
on
Tue Apr 01 19:40:57 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
05Q5D4BAWY
|
| Record Status |
Validated (UNII)
|
| Record Version |
|
-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
|
Common Name | English | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
|
481211-26-1
Created by
admin on Tue Apr 01 19:40:57 GMT 2025 , Edited by admin on Tue Apr 01 19:40:57 GMT 2025
|
PRIMARY | |||
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P51449
Created by
admin on Tue Apr 01 19:40:57 GMT 2025 , Edited by admin on Tue Apr 01 19:40:57 GMT 2025
|
PRIMARY | |||
|
RAR-related orphan receptor gamma
Created by
admin on Tue Apr 01 19:40:57 GMT 2025 , Edited by admin on Tue Apr 01 19:40:57 GMT 2025
|
PRIMARY | |||
|
05Q5D4BAWY
Created by
admin on Tue Apr 01 19:40:57 GMT 2025 , Edited by admin on Tue Apr 01 19:40:57 GMT 2025
|
PRIMARY |
| Linkage Type | Residue Index | |||
|---|---|---|---|---|
| COORDINATION COMPOUND | 1_46 | 1_52 | 1_65 | 1_70 |
| COORDINATION COMPOUND | 1_10 | 1_13 | 1_27 |
| Related Record | Type | Details | ||
|---|---|---|---|---|
|
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INHIBITOR -> TARGET |
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||
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INVERSE AGONIST->TARGET |
EC50
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INHIBITOR -> TARGET |
Reduces IL-17 production.
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INHIBITOR -> TARGET |
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INVERSE AGONIST->TARGET |
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INVERSE AGONIST->TARGET |
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Structural Modifications
| Modification Type | Location Site | Location Type | Residue Modified | Extent | Fragment Name | Fragment Approval |
|---|---|---|---|---|---|---|
| AMINO_ACID_SUBSTITUTION | [1_10] [1_13] [1_27] [1_30] | SITE_SPECIFIC | C4-TYPE ZINC FINGER | C56TF4V7OP | ||
| AMINO_ACID_SUBSTITUTION | [1_46] [1_52] [1_62] [1_65] | SITE_SPECIFIC | C4-TYPE ZINC FINGER | C56TF4V7OP |
| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:NUMBER AVERAGE(CALCULATED) | CHEMICAL |
|
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| Molecular Formula | CHEMICAL |
|