U.S. Department of Health & Human Services Divider Arrow National Institutes of Health Divider Arrow NCATS

Approval Year

Substance Class Protein
Created
by admin
on Tue Apr 01 18:21:49 GMT 2025
Edited
by admin
on Tue Apr 01 18:21:49 GMT 2025
Protein Type ENZYME
Protein Sub Type SERINE/THREONINE-PROTEIN KINASE
Sequence Origin HUMAN
Sequence Type COMPLETE
Record UNII
0572XI7C9L
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
CKI-DELTA
Preferred Name English
CASEIN KINASE I ISOFORM DELTA
Common Name English
CSNK1D
Common Name English
CKID
Common Name English
TAU-PROTEIN KINASE CSNK1D
Common Name English
Code System Code Type Description
CAS
1418269-69-8
Created by admin on Tue Apr 01 18:21:49 GMT 2025 , Edited by admin on Tue Apr 01 18:21:49 GMT 2025
NO STRUCTURE GIVEN
EC (ENZYME CLASS)
EC 2.7.11.1
Created by admin on Tue Apr 01 18:21:49 GMT 2025 , Edited by admin on Tue Apr 01 18:21:49 GMT 2025
PRIMARY
EC (ENZYME CLASS)
EC 2.7.11.26
Created by admin on Tue Apr 01 18:21:49 GMT 2025 , Edited by admin on Tue Apr 01 18:21:49 GMT 2025
ALTERNATIVE
FDA UNII
0572XI7C9L
Created by admin on Tue Apr 01 18:21:49 GMT 2025 , Edited by admin on Tue Apr 01 18:21:49 GMT 2025
PRIMARY
UNIPROT
P48730
Created by admin on Tue Apr 01 18:21:49 GMT 2025 , Edited by admin on Tue Apr 01 18:21:49 GMT 2025
PRIMARY
Related Record Type Details
INHIBITOR -> TARGET
Kd
INHIBITOR -> TARGET
Inhibits TDP-43 hyperphosphorylation
IC50

Structural Modifications

Modification Type Location Site Location Type Residue Modified Extent Fragment Name Fragment Approval
AMINO ACID SUBSTITUTION [1_331] [1_370] [1_382] [1_383] [1_384] [1_411] DEXFOSFOSERINE VI4F0K069V
Name Property Type Amount Referenced Substance Defining Parameters References
Molecular Formula CHEMICAL
MOL_WEIGHT CHEMICAL