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Details

Stereochemistry ACHIRAL
Molecular Formula C11H12F3NO.ClH
Molecular Weight 267.675
Optical Activity ( + / - )
Defined Stereocenters 0 / 1
E/Z Centers 0
Charge 0

SHOW SMILES / InChI
Structure of FLUMEXADOL HCL

SMILES

Cl.FC(F)(F)C1=CC(=CC=C1)C2CNCCO2

InChI

InChIKey=KXLNFFBTSVJQCR-UHFFFAOYSA-N
InChI=1S/C11H12F3NO.ClH/c12-11(13,14)9-3-1-2-8(6-9)10-7-15-4-5-16-10;/h1-3,6,10,15H,4-5,7H2;1H

HIDE SMILES / InChI

Molecular Formula C11H12F3NO
Molecular Weight 231.2143
Charge 0
Count
Stereochemistry RACEMIC
Additional Stereochemistry No
Defined Stereocenters 0 / 1
E/Z Centers 0
Optical Activity ( + / - )

Molecular Formula ClH
Molecular Weight 36.461
Charge 0
Count
Stereochemistry ACHIRAL
Additional Stereochemistry No
Defined Stereocenters 0 / 0
E/Z Centers 0
Optical Activity NONE

FLUMEXADOL is a non-opioid analgesic. Its prodrug OXAFLOZANE was used as an antidepressant in France till 2004.

Approval Year

PubMed

PubMed

TitleDatePubMed
Metabolites of 2-(3-trifluoromethylphenyl)tetrahydro-1,4-oxazine (CERM) 1841) in rats and dogs.
1979-11
The pharmacology of 1841 CERM, a new analgesic.
1978
Substance Class Chemical
Created
by admin
on Tue Apr 01 20:17:16 GMT 2025
Edited
by admin
on Tue Apr 01 20:17:16 GMT 2025
Record UNII
051LY093UV
Record Status Validated (UNII)
Record Version
  • Download
Name Type Language
FLUMEXADOL HCL
Common Name English
NSC-315283
Preferred Name English
Code System Code Type Description
CAS
31599-68-5
Created by admin on Tue Apr 01 20:17:16 GMT 2025 , Edited by admin on Tue Apr 01 20:17:16 GMT 2025
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PUBCHEM
208046
Created by admin on Tue Apr 01 20:17:16 GMT 2025 , Edited by admin on Tue Apr 01 20:17:16 GMT 2025
PRIMARY
FDA UNII
051LY093UV
Created by admin on Tue Apr 01 20:17:16 GMT 2025 , Edited by admin on Tue Apr 01 20:17:16 GMT 2025
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NSC
315283
Created by admin on Tue Apr 01 20:17:16 GMT 2025 , Edited by admin on Tue Apr 01 20:17:16 GMT 2025
PRIMARY