Approval Year
| Substance Class |
Protein
Created
by
admin
on
Edited
Mon Mar 31 22:55:20 GMT 2025
by
admin
on
Mon Mar 31 22:55:20 GMT 2025
|
| Protein Sub Type | |
| Sequence Type | COMPLETE |
| Record UNII |
042A8N37WH
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| Record Status |
Validated (UNII)
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| Record Version |
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-
Download
| Name | Type | Language | ||
|---|---|---|---|---|
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Common Name | English | ||
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Preferred Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English | ||
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Common Name | English |
| Code System | Code | Type | Description | ||
|---|---|---|---|---|---|
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64647
Created by
admin on Mon Mar 31 22:55:20 GMT 2025 , Edited by admin on Mon Mar 31 22:55:20 GMT 2025
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PRIMARY | |||
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042A8N37WH
Created by
admin on Mon Mar 31 22:55:20 GMT 2025 , Edited by admin on Mon Mar 31 22:55:20 GMT 2025
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PRIMARY | |||
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57339251
Created by
admin on Mon Mar 31 22:55:20 GMT 2025 , Edited by admin on Mon Mar 31 22:55:20 GMT 2025
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PRIMARY | |||
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m1878
Created by
admin on Mon Mar 31 22:55:20 GMT 2025 , Edited by admin on Mon Mar 31 22:55:20 GMT 2025
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PRIMARY | Merck Index | ||
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DTXSID70856172
Created by
admin on Mon Mar 31 22:55:20 GMT 2025 , Edited by admin on Mon Mar 31 22:55:20 GMT 2025
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PRIMARY | |||
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107761-42-2
Created by
admin on Mon Mar 31 22:55:20 GMT 2025 , Edited by admin on Mon Mar 31 22:55:20 GMT 2025
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PRIMARY |
| Related Record | Type | Details | ||
|---|---|---|---|---|
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INHIBITOR OF AGGREGATION->TARGET |
A? was maintained in a random-coil/?-helical rich conformation in the presence of Tramiprosate at a 20:1 ratio of Tramiprosate:A?. Binds and shows anti-fibrillogenic activity.
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VACCINE ANTIGEN->TARGET |
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LIGAND->TARGET |
Targets soluble A? monomer to shift oligomer equilibrium and prevent direct neurotoxicity from soluble forms.
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INHIBITOR OF RELEASE->TARGET |
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RADIOLIGAND->TARGET |
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LIGAND->TARGET |
Designed to increase the clearance from the brain of soluble A?, peptides that may lead to toxic effects in the synapses and precede the deposition of fibrillary amyloid.
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INHIBITOR -> TARGET | |||
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RADIOLIGAND->TARGET |
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INHIBITOR OF AGGREGATION->TARGET |
Inhibitor of neuroinflammation caused by A?1–42-induced macrophage production of nitric oxide, TNF-alpha, IL-1beta, and IL-6.
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| Name | Property Type | Amount | Referenced Substance | Defining | Parameters | References |
|---|---|---|---|---|---|---|
| MOL_WEIGHT:SEQUENCE(CALCULATED) | CHEMICAL |
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| Molecular Formula | CHEMICAL |
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