AR-C-239

COC1=CC=CC=C1N2CCN(CCN3C(=O)C4=CC=CC=C4C(C)(C)C3=O)CC2

InChIKey=JFNKXGOEOQCXDM-UHFFFAOYSA-N

InChI=1S/C24H29N3O3/c1-24(2)19-9-5-4-8-18(19)22(28)27(23(24)29)17-14-25-12-15-26(16-13-25)20-10-6-7-11-21(20)30-3/h4-11H,12-17H2,1-3H3

Targets

Primary Target	Pharmacology	Condition	Potency
Alpha-2b adrenergic receptor 35 Target ID: CHEMBL1942 Sources: https://www.ncbi.nlm.nih.gov/pubmed/6171685	Antagonist 2849		8.8 null [pKd]
Alpha-2a adrenergic receptor 70 Target ID: CHEMBL1867 Sources: https://www.ncbi.nlm.nih.gov/pubmed/2835476	Antagonist 2849		6.7 null [pKd]

Name

Type

Language

AR-C-239

Common Name

English

AR-C239

Preferred Name

English

1,3(2H,4H)-ISOQUINOLINEDIONE, 2-(2-(4-(2-METHOXYPHENYL)-1-PIPERAZINYL)ETHYL)-4,4-DIMETHYL-

Systematic Name

English

ARC-239

Code

English

Code System Code Type Description

FDA UNII

M7H349ZZ5T

Created by admin on Mon Mar 31 19:01:24 GMT 2025 , Edited by admin on Mon Mar 31 19:01:24 GMT 2025

PRIMARY

PUBCHEM

609483

Created by admin on Mon Mar 31 19:01:24 GMT 2025 , Edited by admin on Mon Mar 31 19:01:24 GMT 2025

PRIMARY

CAS

67339-62-2

Created by admin on Mon Mar 31 19:01:24 GMT 2025 , Edited by admin on Mon Mar 31 19:01:24 GMT 2025

PRIMARY

EPA CompTox

DTXSID70986600

Created by admin on Mon Mar 31 19:01:24 GMT 2025 , Edited by admin on Mon Mar 31 19:01:24 GMT 2025

PRIMARY

ACTIVE MOIETY


					M7H349ZZ5T

AR-C-239