ALLYLPRODINE

U.S. Department of Health & Human Services Divider Arrow

National Institutes of Health Divider Arrow

NCATS

Description
Sources: https://www.ncbi.nlm.nih.gov/pubmed/13412197 | https://www.ncbi.nlm.nih.gov/pubmed/1246054 | https://www.deadiversion.usdoj.gov/fed_regs/quotas/2014/fr0825.htm

Allylprodine (Ro 2-7113) is an opioid analgesic. It is stereoselective, with one isomer being much more active. Allylprodine is included in Schedule I of the US Controlled Substances Act 1970 as a Narcotic with ACSCN 9602 and a 2014 annual aggregate manufacturing quota of 2 grammes.

Originator

Approval Year

PubMed

PubMed

Title	Date	PubMed
Analgesic activity and toxicity of Ro 2-7113.	1957 Jan 1	13412197
Stereochemical studies on medicinal agents. 19. X-ray crystal structures of two (+/-)-allylprodine diastereomers. The role of the allyl group in conferring high stereoselectivity and potency at analgetic receptors.	1976 Jan	1246054
Conformation of 2,9-dimethyl-3'-hydroxy-5-phenyl-6,7-genzomorphan and its relation to other analgetics and enkephalin.	1978 Jul	209186
Allylprodine analogues as receptor probes. Evidence that phenolic and nonphenolic ligands interact with different subsites on identical opioid receptors.	1981 Jul	6268787

Patents

Patents

Name

Type

Language

ALLYLPRODINE

Official Name

English

3-ALLYL-1-METHYL-4-PHENYL-4-PROPIONYLOXYPIPERIDINE

Common Name

English

ACSCN-9602

Code

English

ALPERIDINE

Common Name

English

allylprodine [INN]

Common Name

English

DEA NO. 9602

Code

English

NIH-7440

Code

English

IDS-NA-007

Code

English

ALLYLPRODINE [MI]

Common Name

English

RO 2-7113

Common Name

English

Classification Tree Code System Code

NCI_THESAURUS

C241

Created by admin on Fri Dec 15 16:05:44 GMT 2023 , Edited by admin on Fri Dec 15 16:05:44 GMT 2023

DEA NO.

9602

Created by admin on Fri Dec 15 16:05:44 GMT 2023 , Edited by admin on Fri Dec 15 16:05:44 GMT 2023

Code System Code Type Description

INN

891

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EPA CompTox

DTXSID80865210

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ChEMBL

CHEMBL2103995

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MERCK INDEX

m1557

Created by admin on Fri Dec 15 16:05:44 GMT 2023 , Edited by admin on Fri Dec 15 16:05:44 GMT 2023

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Merck Index

NCI_THESAURUS

C72102

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DRUG BANK

DB01542

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PUBCHEM

32938

Created by admin on Fri Dec 15 16:05:44 GMT 2023 , Edited by admin on Fri Dec 15 16:05:44 GMT 2023

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FDA UNII

4343OEZ18O

Created by admin on Fri Dec 15 16:05:44 GMT 2023 , Edited by admin on Fri Dec 15 16:05:44 GMT 2023

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WIKIPEDIA

ALLYLPRODINE

Created by admin on Fri Dec 15 16:05:44 GMT 2023 , Edited by admin on Fri Dec 15 16:05:44 GMT 2023

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CAS

25384-17-2

Created by admin on Fri Dec 15 16:05:44 GMT 2023 , Edited by admin on Fri Dec 15 16:05:44 GMT 2023

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EVMPD

SUB05340MIG

Created by admin on Fri Dec 15 16:05:44 GMT 2023 , Edited by admin on Fri Dec 15 16:05:44 GMT 2023

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All of the following components must be present:


					G98M360H09

ALLYLPRODINE, .ALPHA.-


					028U1A6J7B

ALLYLPRODINE, .BETA.-

ACTIVE MOIETY


					4343OEZ18O

SALT/SOLVATE (PARENT)


					WF82M29MCG

ALLYLPRODINE HYDROCHLORIDE, .BETA.-

Definition References