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ALLYLPRODINE
4343OEZ18O
Investigational
ALLYLPRODINE
4343OEZ18O
Investigational
Description
Allylprodine (Ro 2-7113) is an opioid analgesic. It is stereoselective, with one isomer being much more active. Allylprodine is included in Schedule I of the US Controlled Substances Act 1970 as a Narcotic with ACSCN 9602 and a 2014 annual aggregate manufacturing quota of 2 grammes.
Stereochemical studies on medicinal agents. 19. X-ray crystal structures of two (+/-)-allylprodine diastereomers. The role of the allyl group in conferring high stereoselectivity and potency at analgetic receptors.
Allylprodine analogues as receptor probes. Evidence that phenolic and nonphenolic ligands interact with different subsites on identical opioid receptors.
